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Assay Detail

CHEMBL815438

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding potency against V1 receptor in rat liver cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Vasopressin V1a receptor (CHEMBL2868)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Preparation and biological activities of potential vasopressin photoaffinity labels.
Barbeau D, Guay S, Neugebauer W, Escher E.
J Med Chem (1992) 35 : 151 -157
PubMed 1732523 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 2 9.26 9.32

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2115364 1 9.32
CHEMBL373742 VASOPRESSIN 4.0 1 9.19

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2115364 Kd = 0.48 nM 9.32
CHEMBL373742 VASOPRESSIN Kd = 0.64 nM 9.19