Vasopressin V1a receptor · SINGLE PROTEIN · Rattus norvegicus
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As of 2026-09-14Protein identity stays anchored to UniProt P30560. Use UniProt P30560 as the stable identity anchor, then attach disease evidence before program review.
Use UniProt P30560 as the stable identity anchor, then attach disease evidence before program review.
Vasopressin V1a receptor
Review this target as Vasopressin V1a receptor, mapped to UniProt P30560. Sequence length is 424 aa.
Protein source · UniProt accession via ChEMBL component mappingKeep the review anchor, source IDs, and context contract aligned before reusing this target elsewhere.
This review treats Vasopressin V1a receptor as ChEMBL target CHEMBL2868, mapped to UniProt P30560. Disease framing currently uses the Open Targets-ready proxy contract.
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| Preferred Name | Vasopressin V1a receptor |
| Target Type | SINGLE PROTEIN |
| Organism | Rattus norvegicus |
| UniProt | P30560 |
Reviewable protein naming and mapping context for this target snapshot.
| Protein Label | Vasopressin V1a receptor |
| UniProt Accession | P30560 |
| Component Type | Protein |
| Sequence Length | 424 aa |
Vasopressin V1a receptor
Review this target as Vasopressin V1a receptor, mapped to UniProt P30560. Sequence length is 424 aa.
| ChEMBL ID | pChEMBL | Type | Value (nM) | Phase |
|---|---|---|---|---|
| CHEMBL405440 | 10.4 | Kd | 0.04 | Preclinical |
| CHEMBL405440 | 10.4 | Ki | 0.04 | Preclinical |
| CHEMBL265048 | 10.27 | Kd | 0.054 | Preclinical |
| CHEMBL373742 | 10.2 | EC50 | 0.0631 | Approved |
| CHEMBL1819441 | 10.15 | EC50 | 0.07 | Preclinical |
| CHEMBL1817706 | 10.0 | EC50 | 0.1 | Preclinical |
| CHEMBL310921 | 9.99 | Ki | 0.102 | Preclinical |
| CHEMBL424905 | 9.96 | Ki | 0.11 | Preclinical |
| CHEMBL1819542 | 9.92 | EC50 | 0.12 | Preclinical |
| CHEMBL412192 | 9.92 | Ki | 0.12 | Preclinical |
| BAO Format | Assays | Compounds | Avg pChEMBL |
|---|---|---|---|
| single protein format | 24 | 89 | 7.4 |
| assay format | 21 | 199 | 6.3 |
| cell-based format | 11 | 51 | 8.0 |
| cell membrane format | 9 | 48 | 7.0 |
| tissue-based format | 4 | 0 | — |
| BAO Format | Assays | Compounds | Avg pChEMBL |
|---|---|---|---|
| organism-based format | 14 | 0 | — |
| tissue-based format | 4 | 4 | 6.9 |
| assay format | 3 | 0 | — |
| cell-based format | 2 | 23 | 9.1 |