Assay Detail
Binding
CHEMBL815439
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of the 3 nM VP stimulation of phospholipase-C in cultured WRK cells was used as a V1-mediated assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Cell Type | WRK |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Preparation and biological activities of potential vasopressin photoaffinity labels.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 8.72 | 8.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2115364 | — | — | 1 | 8.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2115364 | — | Ki | = | 1.9 | nM | 8.72 |