Assay Detail
Functional
CHEMBL815574
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonistic activity against Tachykinin receptor 3 was determined in the rat everted portal vein (RPV)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Conformational analysis of three NK1 tripeptide antagonists: a proton nuclear magnetic resonance study.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 5.40 | 5.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL156186 | — | — | 1 | 5.80 |
| CHEMBL157858 | — | — | 1 | 5.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL156186 | — | Kd | = | 1584.89 | nM | 5.80 |
| CHEMBL157858 | — | Kd | = | 10000.0 | nM | 5.00 |