Assay Detail
Binding
CHEMBL815745
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Binding affinity towards human Urotensin 2 receptor was determined
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Unraveling the active conformation of urotensin II.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 5 | 9.04 | 9.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL390094 | — | — | 1 | 9.70 |
| CHEMBL426020 | — | — | 1 | 9.60 |
| CHEMBL437430 | HUMAN UROTENSIN II | — | 1 | 9.10 |
| CHEMBL2370836 | — | — | 1 | 8.90 |
| CHEMBL2372643 | — | — | 1 | 7.90 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL390094 | — | Ki | = | 0.1995 | nM | 9.70 |
| CHEMBL426020 | — | Ki | = | 0.2512 | nM | 9.60 |
| CHEMBL437430 | HUMAN UROTENSIN II | Ki | = | 0.7943 | nM | 9.10 |
| CHEMBL2370836 | — | Ki | = | 1.259 | nM | 8.90 |
| CHEMBL2372643 | — | Ki | = | 12.59 | nM | 7.90 |