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Assay Detail

CHEMBL816379

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
The effective concentration to show 50% of activity was measured on varicella zoster virus(VZV) cell culture
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human alphaherpesvirus 3
Confidence 1 — Organism
Curated By Intermediate

Target

Human alphaherpesvirus 3 (CHEMBL613132)
Type ORGANISM
Organism Human alphaherpesvirus 3

Publication

Structure-activity relationships of (E)-5-(2-bromovinyl)uracil and related pyrimidine nucleosides as antiviral agents for herpes viruses.
Choi Y, Li L, Grill S, Gullen E, Lee CS, Gumina G, Tsujii E, Cheng YC, Chu CK.
J Med Chem (2000) 43 : 2538 -2546
PubMed 10891113 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 5.81 6.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1540 PENCICLOVIR 4.0 1 6.85
CHEMBL85809 1 4.77

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1540 PENCICLOVIR EC50 = 140.0 nM 6.85
CHEMBL85809 EC50 = 17000.0 nM 4.77