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Assay Detail

CHEMBL817574

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Compound was tested for inhibition of trypsin
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Bos taurus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Serine protease 1 (CHEMBL3769)
Type SINGLE PROTEIN
Organism Bos taurus

Publication

3-Amidinophenylalanine-based inhibitors of urokinase.
Stürzebecher J, Vieweg H, Steinmetzer T, Schweinitz A, Stubbs MT, Renatus M, Wikström P.
Bioorg Med Chem Lett (1999) 9 : 3147 -3152
PubMed 10560742 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.43 7.43

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL107955 1 7.43

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL107955 Ki = 37.0 nM 7.43