Assay Detail
Binding
CHEMBL818262
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Compound was evaluated for its inhibitory activity against bovine pancreatic trypsin
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bos taurus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Inhibition of serine proteases: activity of 1,3-diazetidine-2,4-diones.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.17 | 7.41 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL47394 | — | — | 1 | 7.41 |
| CHEMBL296771 | — | — | 1 | 6.70 |
| CHEMBL298276 | — | — | 1 | 4.41 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL47394 | — | IC50 | = | 39.0 | nM | 7.41 |
| CHEMBL296771 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL298276 | — | IC50 | = | 39000.0 | nM | 4.41 |