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Assay Detail

CHEMBL820107

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity evaluated against Varicella Zoster virus (YS)
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human alphaherpesvirus 3
Confidence 1 — Organism
Curated By Intermediate

Target

Human alphaherpesvirus 3 (CHEMBL613132)
Type ORGANISM
Organism Human alphaherpesvirus 3

Publication

Novel bicyclic furanopyrimidines with dual anti-VZV and -HCMV activity.
McGuigan C, Brancale A, Andrei G, Snoeck R, De Clercq E, Balzarini J.
Bioorg Med Chem Lett (2003) 13 : 4511 -4513
PubMed 14643358 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 7.44 7.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3143173 1 7.70
CHEMBL3143172 1 7.52
CHEMBL3143167 1 7.52
CHEMBL3143171 1 7.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3143173 EC50 = 20.0 nM 7.70
CHEMBL3143172 EC50 = 30.0 nM 7.52
CHEMBL3143167 EC50 = 30.0 nM 7.52
CHEMBL3143171 EC50 = 100.0 nM 7.00