Assay Detail
Binding
CHEMBL822646
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]PDBU from protein kinase C-alpha
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Synthesis of ingenol analogs wth affinity for protein kinase C
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 8.32 | 9.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL46094 | — | — | 1 | 9.85 |
| CHEMBL156719 | — | — | 1 | 6.78 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL46094 | — | Ki | = | 0.14 | nM | 9.85 |
| CHEMBL156719 | — | Ki | = | 165.0 | nM | 6.78 |