Assay Detail
Binding
CHEMBL822796
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Binding potency for nAChR subtype Alpha-1-beta-1-delta gamma(torpedo)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Torpedo |
| Confidence | 6 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Neuronal nicotinic acetylcholine receptors as targets for drug discovery.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 7.54 | 8.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL6623 | EPIBATIDINE | — | 1 | 8.57 |
| CHEMBL335712 | — | — | 1 | 6.50 |
| CHEMBL274525 | ABT-418 | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL6623 | EPIBATIDINE | Ki | = | 2.7 | nM | 8.57 |
| CHEMBL335712 | — | Ki | = | 314.0 | nM | 6.50 |
| CHEMBL274525 | ABT-418 | Ki | > | 10000.0 | nM | - |