Assay Detail

CHEMBL824914

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional

Inhibitory concentration measured against the prostate cancer cell line DU145

ChEMBL ↗

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Target

NON-PROTEIN TARGET (CHEMBL3879801) ↗

Open DB target context

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Primary target NON-PROTEIN TARGET

CHEMBL3879801

Anchored from Assay target.

Protein identity NON-PROTEIN TARGET

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Functional
Organism	Homo sapiens
Cell Type	Cancer cell lines
Confidence	1 — Organism
Curated By	Autocuration

Target

NON-PROTEIN TARGET (CHEMBL3879801) ↗

Type	NON-MOLECULAR

Publication

Truncated azinomycin analogues intercalate into DNA.

Casely-Hayford MA, Pors K, Patterson LH, Gerner C, Neidle S, Searcey M.
Bioorg Med Chem Lett (2005) 15 : 653 -656
PubMed 15664831 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
IC50	1	7.30	7.30

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL78703	—	—	1	7.30

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL78703	—	IC50	=	50.0	nM	7.30