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Assay Detail

CHEMBL826401

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibitory concentration against MeVo melanoma cell line
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Confidence 1 — Organism
Curated By Autocuration

Publication

Synthesis and cytotoxic evaluation of novel spirohydantoin derivatives of the dihydrothieno[2,3-b]naphtho-4,9-dione system.
Gomez-Monterrey I, Santelli G, Campiglia P, Califano D, Falasconi F, Pisano C, Vesci L, Lama T, Grieco P, Novellino E.
J Med Chem (2005) 48 : 1152 -1157
PubMed 15715481 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 6.35 6.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL178282 1 6.60
CHEMBL53463 DOXORUBICIN 4.0 1 6.09

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL178282 IC50 = 250.0 nM 6.60
CHEMBL53463 DOXORUBICIN IC50 = 820.0 nM 6.09