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Assay Detail

CHEMBL826577

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Functional
Potency of compound in glycogen accumulation in L6 cells
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Rattus norvegicus
Cell Type L6
Confidence 1 — Organism
Curated By Intermediate

Target

L6 (CHEMBL614793)
Type CELL-LINE
Organism Rattus norvegicus

Publication

4-Acylamino-6-arylfuro[2,3-d]pyrimidines: potent and selective glycogen synthase kinase-3 inhibitors.
Maeda Y, Nakano M, Sato H, Miyazaki Y, Schweiker SL, Smith JL, Truesdale AT.
Bioorg Med Chem Lett (2004) 14 : 3907 -3911
PubMed 15225695 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 3 6.27 6.41

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL182419 1 6.41
CHEMBL361196 1 6.13
CHEMBL183038 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL182419 EC50 = 390.0 nM 6.41
CHEMBL361196 EC50 = 740.0 nM 6.13
CHEMBL183038 EC50 > 10000.0 nM -