Assay Detail
Binding
CHEMBL826982
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Dissociation constant for ERK2 kinase
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Identification of novel extracellular signal-regulated kinase docking domain inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 3 | 5.13 | 5.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL364953 | — | — | 1 | 5.30 |
| CHEMBL363555 | — | — | 1 | 5.30 |
| CHEMBL190710 | — | — | 1 | 4.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL364953 | — | Kd | = | 5000.0 | nM | 5.30 |
| CHEMBL363555 | — | Kd | = | 5000.0 | nM | 5.30 |
| CHEMBL190710 | — | Kd | = | 16000.0 | nM | 4.80 |