Assay Detail
Binding
CHEMBL828218
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity for fatty acid amide hydrolase
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
The endocannabinoid system: drug targets, lead compounds, and potential therapeutic applications.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 5 | 8.44 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL371831 | — | — | 1 | 9.00 |
| CHEMBL422064 | — | — | 1 | 8.92 |
| CHEMBL35925 | — | — | 1 | 8.64 |
| CHEMBL191424 | — | — | 1 | 8.04 |
| CHEMBL91417 | — | — | 1 | 7.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL371831 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL422064 | — | Ki | = | 1.2 | nM | 8.92 |
| CHEMBL35925 | — | Ki | = | 2.3 | nM | 8.64 |
| CHEMBL191424 | — | Ki | = | 9.1 | nM | 8.04 |
| CHEMBL91417 | — | Ki | = | 25.0 | nM | 7.60 |