Assay Detail
Binding
CHEMBL828732
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Inhibition of putrescine binding to Pea seedling amine oxidase
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Pisum sativum |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Alkylamino derivatives of 4-aminomethylpyridine as inhibitors of copper-containing amine oxidases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 7 | 4.53 | 5.03 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL537624 | — | — | 1 | 5.03 |
| CHEMBL534467 | — | — | 1 | 4.77 |
| CHEMBL537623 | — | — | 1 | 4.26 |
| CHEMBL541126 | — | — | 1 | 4.05 |
| CHEMBL537628 | — | — | 1 | - |
| CHEMBL536949 | — | — | 1 | - |
| CHEMBL537401 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL537624 | — | IC50 | = | 9300.0 | nM | 5.03 |
| CHEMBL534467 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL537623 | — | IC50 | = | 55000.0 | nM | 4.26 |
| CHEMBL541126 | — | IC50 | = | 89000.0 | nM | 4.05 |
| CHEMBL537628 | — | IC50 | = | 1000000.0 | nM | - |
| CHEMBL536949 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL537401 | — | IC50 | = | 330000.0 | nM | - |