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Assay Detail

CHEMBL828869

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity for aryl hydrocarbon receptor (AhR) of rabbit liver cytosol incubated with 0.2 nM [3H]-TCDD; Agonist
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Oryctolagus cuniculus
Tissue Liver
Subcellular Cytosol
Confidence 9 — Direct single protein target
Curated By Expert

Target

Aryl hydrocarbon receptor (CHEMBL4725)
Type SINGLE PROTEIN
Organism Oryctolagus cuniculus

Publication

Synthesis and biological properties of new stilbene derivatives of resveratrol as new selective aryl hydrocarbon modulators.
de Medina P, Casper R, Savouret JF, Poirot M.
J Med Chem (2005) 48 : 287 -291
PubMed 15634023 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 9.70 9.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL179510 1 9.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL179510 Ki = 0.2 nM 9.70