Assay Detail
Binding
CHEMBL829692
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity for adenosine A1 receptor by using as [3H]CPX radioligand in membranes from Chinese hamster ovary cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | ovary |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
The discovery of a selective, high affinity A(2B) adenosine receptor antagonist for the potential treatment of asthma.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 8.10 | 8.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL178172 | — | — | 1 | 8.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL178172 | — | Ki | = | 8.0 | nM | 8.10 |