Assay Detail
Binding
CHEMBL829880
Review assay metadata, readout intent, target linkage, and publication context from the same page.
In vitro effective concentration for mouse corticotropin releasing factor 2 receptor
55
Total Activities
55
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Target
Corticotropin-releasing factor receptor 2 (CHEMBL2253) ↗| Type | SINGLE PROTEIN |
| Organism | Mus musculus |
Publication
Discovery of corticotropin releasing factor 2 receptor selective sauvagine analogues for treatment of skeletal muscle atrophy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 55 | 8.00 | 8.74 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL437089 | — | — | 1 | 8.74 |
| CHEMBL267635 | — | — | 1 | 8.72 |
| CHEMBL413414 | — | — | 1 | 8.52 |
| CHEMBL411590 | — | — | 1 | 8.48 |
| CHEMBL438220 | — | — | 1 | 8.40 |
| CHEMBL438948 | — | — | 1 | 8.39 |
| CHEMBL412026 | — | — | 1 | 8.37 |
| CHEMBL429970 | HUMAN UROCORTIN 2 | — | 1 | 8.37 |
| CHEMBL430078 | — | — | 1 | 8.33 |
| CHEMBL410347 | — | — | 1 | 8.32 |
| CHEMBL427923 | — | — | 1 | 8.30 |
| CHEMBL264275 | — | — | 1 | 8.30 |
| CHEMBL438939 | — | — | 1 | 8.28 |
| CHEMBL438601 | — | — | 1 | 8.26 |
| CHEMBL438928 | — | — | 1 | 8.25 |
| CHEMBL427811 | — | — | 1 | 8.25 |
| CHEMBL428824 | — | — | 1 | 8.24 |
| CHEMBL436914 | — | — | 1 | 8.23 |
| CHEMBL409748 | — | — | 1 | 8.19 |
| CHEMBL442112 | — | — | 1 | 8.15 |
| CHEMBL438391 | — | — | 1 | 8.14 |
| CHEMBL414130 | — | — | 1 | 8.13 |
| CHEMBL436912 | — | — | 1 | 8.11 |
| CHEMBL268549 | — | — | 1 | 8.07 |
| CHEMBL415130 | — | — | 1 | 8.07 |
| CHEMBL437289 | — | — | 1 | 8.07 |
| CHEMBL410568 | — | — | 1 | 8.06 |
| CHEMBL428809 | — | — | 1 | 8.03 |
| CHEMBL263862 | — | — | 1 | 8.00 |
| CHEMBL429403 | — | — | 1 | 7.97 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL437089 | — | EC50 | = | 1.8 | nM | 8.74 |
| CHEMBL267635 | — | EC50 | = | 1.9 | nM | 8.72 |
| CHEMBL413414 | — | EC50 | = | 3.0 | nM | 8.52 |
| CHEMBL411590 | — | EC50 | = | 3.3 | nM | 8.48 |
| CHEMBL438220 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL438948 | — | EC50 | = | 4.1 | nM | 8.39 |
| CHEMBL412026 | — | EC50 | = | 4.3 | nM | 8.37 |
| CHEMBL429970 | HUMAN UROCORTIN 2 | EC50 | = | 4.3 | nM | 8.37 |
| CHEMBL430078 | — | EC50 | = | 4.7 | nM | 8.33 |
| CHEMBL410347 | — | EC50 | = | 4.8 | nM | 8.32 |
| CHEMBL427923 | — | EC50 | = | 5.0 | nM | 8.30 |
| CHEMBL264275 | — | EC50 | = | 5.0 | nM | 8.30 |
| CHEMBL438939 | — | EC50 | = | 5.2 | nM | 8.28 |
| CHEMBL438601 | — | EC50 | = | 5.5 | nM | 8.26 |
| CHEMBL427811 | — | EC50 | = | 5.6 | nM | 8.25 |
| CHEMBL438928 | — | EC50 | = | 5.6 | nM | 8.25 |
| CHEMBL428824 | — | EC50 | = | 5.8 | nM | 8.24 |
| CHEMBL436914 | — | EC50 | = | 5.9 | nM | 8.23 |
| CHEMBL409748 | — | EC50 | = | 6.5 | nM | 8.19 |
| CHEMBL442112 | — | EC50 | = | 7.0 | nM | 8.15 |
| CHEMBL438391 | — | EC50 | = | 7.2 | nM | 8.14 |
| CHEMBL414130 | — | EC50 | = | 7.4 | nM | 8.13 |
| CHEMBL436912 | — | EC50 | = | 7.8 | nM | 8.11 |
| CHEMBL437289 | — | EC50 | = | 8.5 | nM | 8.07 |
| CHEMBL268549 | — | EC50 | = | 8.6 | nM | 8.07 |
| CHEMBL415130 | — | EC50 | = | 8.5 | nM | 8.07 |
| CHEMBL410568 | — | EC50 | = | 8.8 | nM | 8.06 |
| CHEMBL428809 | — | EC50 | = | 9.4 | nM | 8.03 |
| CHEMBL263862 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL429403 | — | EC50 | = | 10.7 | nM | 7.97 |
| CHEMBL414711 | — | EC50 | = | 10.9 | nM | 7.96 |
| CHEMBL439102 | — | EC50 | = | 12.8 | nM | 7.89 |
| CHEMBL410814 | — | EC50 | = | 13.3 | nM | 7.88 |
| CHEMBL427611 | — | EC50 | = | 14.1 | nM | 7.85 |
| CHEMBL441564 | — | EC50 | = | 14.8 | nM | 7.83 |
| CHEMBL414568 | — | EC50 | = | 15.2 | nM | 7.82 |
| CHEMBL428975 | — | EC50 | = | 15.6 | nM | 7.81 |
| CHEMBL438210 | — | EC50 | = | 16.1 | nM | 7.79 |
| CHEMBL429243 | — | EC50 | = | 18.2 | nM | 7.74 |
| CHEMBL441929 | — | EC50 | = | 19.2 | nM | 7.72 |
| CHEMBL439887 | — | EC50 | = | 19.1 | nM | 7.72 |
| CHEMBL429719 | — | EC50 | = | 20.2 | nM | 7.70 |
| CHEMBL409626 | — | EC50 | = | 20.6 | nM | 7.69 |
| CHEMBL412296 | — | EC50 | = | 21.6 | nM | 7.67 |
| CHEMBL428127 | — | EC50 | = | 21.6 | nM | 7.67 |
| CHEMBL427792 | — | EC50 | = | 21.3 | nM | 7.67 |
| CHEMBL429069 | — | EC50 | = | 21.7 | nM | 7.66 |
| CHEMBL411961 | — | EC50 | = | 22.3 | nM | 7.65 |
| CHEMBL429547 | — | EC50 | = | 23.4 | nM | 7.63 |
| CHEMBL411474 | — | EC50 | = | 24.6 | nM | 7.61 |