Assay Detail
Binding
CHEMBL829951
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cells
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Potent bombesin-like peptides for GRP-receptor targeting of tumors with 99mTc: a preclinical study.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 5 | 8.70 | 9.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL414307 | — | — | 1 | 9.05 |
| CHEMBL413893 | UNIVERSAL LIGAND | — | 1 | 9.02 |
| CHEMBL2371725 | Demobesin 3 | — | 1 | 8.80 |
| CHEMBL266079 | — | — | 1 | 8.70 |
| CHEMBL2371724 | — | — | 1 | 7.95 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL414307 | — | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL413893 | UNIVERSAL LIGAND | IC50 | = | 0.96 | nM | 9.02 |
| CHEMBL2371725 | Demobesin 3 | IC50 | = | 1.6 | nM | 8.80 |
| CHEMBL266079 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL2371724 | — | IC50 | = | 11.2 | nM | 7.95 |