Assay Detail
Binding
CHEMBL830208
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In vitro inhibitory activity towards human cannabinoid receptors 2 using fluorescence assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Chemical modification of the naphthoyl 3-position of JWH-015: in search of a fluorescent probe to the cannabinoid CB2 receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 6.85 | 7.44 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL306764 | — | — | 1 | 7.44 |
| CHEMBL178918 | — | — | 1 | 6.84 |
| CHEMBL368432 | — | — | 1 | 6.72 |
| CHEMBL555145 | — | — | 1 | 6.38 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL306764 | — | Ki | = | 36.0 | nM | 7.44 |
| CHEMBL178918 | — | Ki | = | 143.0 | nM | 6.84 |
| CHEMBL368432 | — | Ki | = | 191.0 | nM | 6.72 |
| CHEMBL555145 | — | Ki | = | 420.0 | nM | 6.38 |