Assay Detail
Binding
CHEMBL830240
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Inhibition constant against human cathepsin H using L-Arg-b-naphthalamide
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Acyclic cyanamide-based inhibitors of cathepsin K.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.34 | 9.34 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL371420 | — | — | 1 | 9.34 |
| CHEMBL189149 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL371420 | — | Ki | = | 0.46 | nM | 9.34 |
| CHEMBL189149 | — | Ki | > | 13000.0 | nM | - |