Assay Detail
Functional
CHEMBL831867
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of calcium mobilization in human eosinophils
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Discovery of CC chemokine receptor-3 (CCR3) antagonists with picomolar potency.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 8.25 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL363840 | — | — | 1 | 9.00 |
| CHEMBL195555 | — | — | 1 | 8.70 |
| CHEMBL382108 | — | — | 1 | 8.70 |
| CHEMBL193575 | — | — | 1 | 8.70 |
| CHEMBL2113074 | — | — | 1 | 8.70 |
| CHEMBL2113077 | — | — | 1 | 8.70 |
| CHEMBL373347 | — | — | 1 | 8.40 |
| CHEMBL365820 | — | — | 1 | 8.40 |
| CHEMBL3706810 | — | — | 1 | 8.40 |
| CHEMBL195433 | — | — | 1 | 8.40 |
| CHEMBL250689 | — | — | 1 | 8.10 |
| CHEMBL175634 | — | — | 1 | 8.00 |
| CHEMBL362466 | — | — | 1 | 7.77 |
| CHEMBL363166 | — | — | 1 | 7.46 |
| CHEMBL193442 | — | — | 1 | 7.30 |
| CHEMBL194141 | — | — | 1 | 7.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL363840 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL195555 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL382108 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL193575 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL2113074 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL2113077 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL373347 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL365820 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL3706810 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL195433 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL250689 | — | IC50 | = | 8.0 | nM | 8.10 |
| CHEMBL175634 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL362466 | — | IC50 | = | 17.0 | nM | 7.77 |
| CHEMBL363166 | — | IC50 | = | 35.0 | nM | 7.46 |
| CHEMBL193442 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL194141 | — | IC50 | = | 50.0 | nM | 7.30 |