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Assay Detail

CHEMBL832401

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibitory concentration against Melatonin receptor type 1B
30
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Expert

Target

Melatonin receptor type 1B (CHEMBL1946)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Tetrahydroisoquinoline derivatives as melatonin MT2 receptor antagonists.
Karageorge GN, Bertenshaw S, Iben L, Xu C, Sarbin N, Gentile A, Dubowchik GM.
Bioorg Med Chem Lett (2004) 14 : 5881 -5884
PubMed 15501061 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 30 7.04 8.26

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL186452 1 8.26
CHEMBL187525 1 8.01
CHEMBL364816 1 8.00
CHEMBL433573 1 7.66
CHEMBL365648 1 7.62
CHEMBL186941 1 7.62
CHEMBL186262 1 7.52
CHEMBL187136 1 7.35
CHEMBL186590 1 7.22
CHEMBL188120 1 7.21
CHEMBL187593 1 7.12
CHEMBL186451 1 7.10
CHEMBL360641 1 7.08
CHEMBL366115 1 7.00
CHEMBL361458 1 6.92
CHEMBL186915 1 6.89
CHEMBL186251 1 6.85
CHEMBL186866 1 6.80
CHEMBL187148 1 6.66
CHEMBL365899 2 6.62
CHEMBL434916 1 6.57
CHEMBL362162 1 6.55
CHEMBL185733 1 6.43
CHEMBL187592 1 6.40
CHEMBL359576 1 6.09
CHEMBL186167 1 6.00
CHEMBL360213 1 -
CHEMBL187016 1 -
CHEMBL364352 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL186452 IC50 = 5.5 nM 8.26
CHEMBL187525 IC50 = 9.7 nM 8.01
CHEMBL364816 IC50 = 9.9 nM 8.00
CHEMBL433573 IC50 = 22.0 nM 7.66
CHEMBL365648 IC50 = 24.0 nM 7.62
CHEMBL186941 IC50 = 24.0 nM 7.62
CHEMBL186262 IC50 = 30.0 nM 7.52
CHEMBL187136 IC50 = 45.0 nM 7.35
CHEMBL186590 IC50 = 60.0 nM 7.22
CHEMBL188120 IC50 = 62.0 nM 7.21
CHEMBL187593 IC50 = 76.0 nM 7.12
CHEMBL186451 IC50 = 79.0 nM 7.10
CHEMBL360641 IC50 = 83.0 nM 7.08
CHEMBL366115 IC50 = 100.0 nM 7.00
CHEMBL361458 IC50 = 120.0 nM 6.92
CHEMBL186915 IC50 = 130.0 nM 6.89
CHEMBL186251 IC50 = 140.0 nM 6.85
CHEMBL186866 IC50 = 160.0 nM 6.80
CHEMBL187148 IC50 = 220.0 nM 6.66
CHEMBL365899 IC50 = 240.0 nM 6.62
CHEMBL434916 IC50 = 270.0 nM 6.57
CHEMBL362162 IC50 = 280.0 nM 6.55
CHEMBL365899 IC50 = 310.0 nM 6.51
CHEMBL185733 IC50 = 370.0 nM 6.43
CHEMBL187592 IC50 = 400.0 nM 6.40
CHEMBL359576 IC50 = 810.0 nM 6.09
CHEMBL186167 IC50 = 1000.0 nM 6.00
CHEMBL187016 IC50 > 1000.0 nM -
CHEMBL360213 IC50 > 1000.0 nM -
CHEMBL364352 IC50 > 1000.0 nM -