Assay Detail
Functional
CHEMBL834806
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Inhibitory concentration was measured against Mel-A (normal melanocyte) cell from mouse at 48 hours
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
N1-substituent effects in the selective delivery of polyamine conjugates into cells containing active polyamine transporters.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.78 | 5.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL541629 | — | — | 1 | 5.08 |
| CHEMBL555288 | — | — | 1 | 4.48 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL541629 | — | IC50 | = | 8300.0 | nM | 5.08 |
| CHEMBL555288 | — | IC50 | = | 32800.0 | nM | 4.48 |