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Assay Detail

CHEMBL838682

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity against alpha-Mannosidase isolated from Jack bean
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Canavalia ensiformis
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Alpha-mannosidase (CHEMBL4193)
Type SINGLE PROTEIN
Organism Glycine max

Publication

Functionalized pyrrolidines inhibit alpha-mannosidase activity and growth of human glioblastoma and melanoma cells.
Fiaux H, Popowycz F, Favre S, Schütz C, Vogel P, Gerber-Lemaire S, Juillerat-Jeanneret L.
J Med Chem (2005) 48 : 4237 -4246
PubMed 15974577 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 2 6.17 7.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL190311 1 7.72
CHEMBL191531 1 4.62

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL190311 Ki = 19.0 nM 7.72
CHEMBL191531 Ki = 24000.0 nM 4.62