Assay Detail
Binding
CHEMBL838698
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity towards Prostaglandin E receptor was determined in rat
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Target
Prostaglandin E2 receptor EP1 subtype (CHEMBL5068) ↗| Type | SINGLE PROTEIN |
| Organism | Rattus norvegicus |
Publication
2,3-Diarylthiophenes as selective EP1 receptor antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.92 | 7.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL362851 | — | — | 1 | 7.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL362851 | — | Ki | = | 12.0 | nM | 7.92 |