Assay Detail
Binding
CHEMBL838702
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Binding affinity for human melanocortin 3 receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Identification of agonists and antagonists of the human melanocortin-4 receptor from piperazinebenzylamines.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.96 | 6.20 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL183799 | — | — | 1 | 6.20 |
| CHEMBL182277 | — | — | 1 | 5.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL183799 | — | Ki | = | 630.0 | nM | 6.20 |
| CHEMBL182277 | — | Ki | = | 1900.0 | nM | 5.72 |