Assay Detail
Binding
CHEMBL838830
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Binding constant for Opioid receptor mu 1 in mouse
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
18F-labeled sufentanil for PET-imaging of mu-opioid receptors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 9.77 | 10.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2311157 | [11C]-CARFENTANIL | 1.0 | 1 | 10.62 |
| CHEMBL196960 | — | — | 1 | 10.00 |
| CHEMBL197479 | — | — | 1 | 8.68 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2311157 | [11C]-CARFENTANIL | Ki | = | 0.024 | nM | 10.62 |
| CHEMBL196960 | — | Ki | = | 0.1 | nM | 10.00 |
| CHEMBL197479 | — | Ki | = | 2.1 | nM | 8.68 |