Assay Detail
Binding
CHEMBL847261
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Enzymatic activity was determined
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Parasite enzymes as potential targets for antiparasitic chemotherapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 4.51 | 4.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL437 | SULFATHIAZOLE | 4.0 | 1 | 4.85 |
| CHEMBL338802 | SULFAGUANIDINE | 4.0 | 1 | 4.16 |
| CHEMBL21 | SULFANILAMIDE | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL437 | SULFATHIAZOLE | Ki | = | 14000.0 | nM | 4.85 |
| CHEMBL338802 | SULFAGUANIDINE | Ki | = | 69000.0 | nM | 4.16 |
| CHEMBL21 | SULFANILAMIDE | Ki | = | 130000.0 | nM | - |