Assay Detail
ADMET
CHEMBL853469
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition at recombinant human CYP2C19
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Discovery of potent CRTh2 (DP2) receptor antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.70 | 5.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL213029 | — | — | 1 | 5.80 |
| CHEMBL209689 | — | — | 1 | 5.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL213029 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL209689 | — | IC50 | = | 2500.0 | nM | 5.60 |