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Assay Detail

CHEMBL853827

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of VZV replication in HFF cells by plaque reduction assay
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human alphaherpesvirus 3
Cell Type HFF
Confidence 1 — Organism
Curated By Expert

Target

Human alphaherpesvirus 3 (CHEMBL613132)
Type ORGANISM
Organism Human alphaherpesvirus 3

Publication

9-{[3-fluoro-2-(hydroxymethyl)cyclopropylidene]methyl}adenines and -guanines. Synthesis and antiviral activity of all stereoisomers1.
Zhou S, Kern ER, Gullen E, Cheng YC, Drach JC, Tamiya S, Mitsuya H, Zemlicka J.
J Med Chem (2006) 49 : 6120 -6128
PubMed 17004726 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 5 4.53 5.23

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL218614 1 5.23
CHEMBL217219 1 4.47
CHEMBL386690 1 4.26
CHEMBL384629 1 4.17
CHEMBL383977 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL218614 EC50 = 5900.0 nM 5.23
CHEMBL217219 EC50 = 33600.0 nM 4.47
CHEMBL386690 EC50 = 54600.0 nM 4.26
CHEMBL384629 EC50 = 68300.0 nM 4.17
CHEMBL383977 EC50 > 100000.0 nM -