Assay Detail
Functional
CHEMBL854189
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Activity at TP receptor assessed as inhibition of U46619-induced platelet aggregation in platelet rich plasma
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Tissue | Plasma |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Identification of an indole series of prostaglandin D2 receptor antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.73 | 5.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL383484 | — | — | 1 | 5.08 |
| CHEMBL207203 | — | — | 1 | 4.37 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL383484 | — | IC50 | = | 8400.0 | nM | 5.08 |
| CHEMBL207203 | — | IC50 | = | 43000.0 | nM | 4.37 |