Assay Detail
Binding
CHEMBL855086
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Inhibition of rabbit liver guanase
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Oryctolagus cuniculus |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Design of inhibitors against guanase: synthesis and biochemical evaluation of analogues of azepinomycin.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 4.49 | 4.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL374469 | — | — | 1 | 4.70 |
| CHEMBL220699 | — | — | 1 | 4.27 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL374469 | — | Ki | = | 20100.0 | nM | 4.70 |
| CHEMBL220699 | — | Ki | = | 53600.0 | nM | 4.27 |