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Assay Detail

CHEMBL855656

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Functional
ABTS radical scavenging activity
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 1 — Organism
Curated By Autocuration

Publication

Free radical scavengers from the medicinal mushroom Inonotus xeranticus and their proposed biogenesis.
Lee IK, Jung JY, Seok SJ, Kim WG, Yun BS.
Bioorg Med Chem Lett (2006) 16 : 5621 -5624
PubMed 16908141 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 5.08 5.55

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL145 CAFFEIC ACID 3.0 1 5.55
CHEMBL222021 PROTOCATECHUALDEHYDE 1 5.30
CHEMBL3989727 VITAMIN E 4.0 1 5.06
CHEMBL448733 METHYLINOSCAVIN D 1 5.06
CHEMBL218276 INOSCAVIN D 1 4.90
CHEMBL218423 PHELLIGRIDIN D 1 4.86
CHEMBL37537 PROTOCATECHUIC ACID 1 4.80

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL145 CAFFEIC ACID IC50 = 2800.0 nM 5.55
CHEMBL222021 PROTOCATECHUALDEHYDE IC50 = 5000.0 nM 5.30
CHEMBL3989727 VITAMIN E IC50 = 8800.0 nM 5.06
CHEMBL448733 METHYLINOSCAVIN D IC50 = 8700.0 nM 5.06
CHEMBL218276 INOSCAVIN D IC50 = 12500.0 nM 4.90
CHEMBL218423 PHELLIGRIDIN D IC50 = 13700.0 nM 4.86
CHEMBL37537 PROTOCATECHUIC ACID IC50 = 15700.0 nM 4.80