Assay Detail
Functional
CHEMBL856233
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Dose-dependent inhibition of SP-induced increases in phosphatidylinositol turnover in UC11 cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | UC11 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Synthesis and sar of 4-(1H-benzimidazole-2-carbonyl)piperidines with dual histamine H1/tachykinin NK1 receptor antagonist activity
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 7.18 | 7.18 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL93556 | — | — | 1 | 7.18 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL93556 | — | Kd | = | 66.07 | nM | 7.18 |