Assay Detail
Binding
CHEMBL857165
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Inhibition of Epidermal growth factor receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Naphthyl ketones: a new class of Janus kinase 3 inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.30 | 5.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL538798 | — | — | 1 | 5.60 |
| CHEMBL154580 | — | — | 1 | 5.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL538798 | — | IC50 | = | 2511.89 | nM | 5.60 |
| CHEMBL154580 | — | IC50 | = | 10000.0 | nM | 5.00 |