Assay Detail
Functional
CHEMBL857244
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity against alpha-1 adrenergic receptor of rat anococcygeus muscle; value ranges from 6.2-6.5
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Synthesis and alpha 2-adrenoceptor antagonist activity of some disulfonamidobenzoquinolizines.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 6.34 | 6.34 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL30419 | — | — | 1 | 6.34 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL30419 | — | Kd | = | 457.09 | nM | 6.34 |