Assay Detail
Binding
CHEMBL857508
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The apparent binding affinity against cathepsin L.
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Protease inhibitors: current status and future prospects.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 6.32 | 6.47 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL281540 | — | — | 1 | 6.47 |
| CHEMBL57836 | — | — | 1 | 6.16 |
| CHEMBL113805 | — | — | 1 | - |
| CHEMBL113724 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL281540 | — | Ki | = | 340.0 | nM | 6.47 |
| CHEMBL57836 | — | Ki | = | 700.0 | nM | 6.16 |
| CHEMBL113805 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL113724 | — | Ki | > | 1000.0 | nM | - |