Assay Detail
Binding
CHEMBL867575
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Inhibitory activity against class I FBP aldolase from rabbit
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Oryctolagus cuniculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Target
Fructose-bisphosphate aldolase A (CHEMBL4695) ↗| Type | SINGLE PROTEIN |
| Organism | Oryctolagus cuniculus |
Publication
N-Sulfonyl hydroxamate derivatives as inhibitors of class II fructose-1,6-diphosphate aldolase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 6 | 6.00 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL371668 | PHOSPHOGLYCOLOHYDROXAMATE | — | 1 | 6.00 |
| CHEMBL196442 | — | — | 1 | - |
| CHEMBL370845 | — | — | 1 | - |
| CHEMBL197860 | — | — | 1 | - |
| CHEMBL202288 | — | — | 1 | - |
| CHEMBL199843 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL371668 | PHOSPHOGLYCOLOHYDROXAMATE | Ki | = | 1000.0 | nM | 6.00 |
| CHEMBL196442 | — | Ki | > | 1000000.0 | nM | - |
| CHEMBL370845 | — | Ki | > | 10000000.0 | nM | - |
| CHEMBL197860 | — | Ki | > | 10000000.0 | nM | - |
| CHEMBL202288 | — | Ki | > | 10000000.0 | nM | - |
| CHEMBL199843 | — | Ki | > | 10000000.0 | nM | - |