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Assay Detail

CHEMBL867772

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of jack beans alpha-mannosidase
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Canavalia ensiformis
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Alpha-mannosidase (CHEMBL4193)
Type SINGLE PROTEIN
Organism Glycine max

Publication

Fluorescent glycosidase inhibiting 1,5-dideoxy-1,5-iminoalditols.
Greimel P, Häusler H, Lundt I, Rupitz K, Stütz AE, Tarling CA, Withers SG, Wrodnigg TM.
Bioorg Med Chem Lett (2006) 16 : 2067 -2070
PubMed 16481162 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 3 4.35 4.75

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL84844 DEOXYMANNOJIRIMYCIN 1 4.75
CHEMBL207481 1 4.19
CHEMBL206357 1 4.11

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL84844 DEOXYMANNOJIRIMYCIN Ki = 18000.0 nM 4.75
CHEMBL207481 Ki = 65000.0 nM 4.19
CHEMBL206357 Ki = 78000.0 nM 4.11