Assay Detail
Functional
CHEMBL867962
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Activity at human FPRL1-mediated calcium mobilization in CHO cells
36
Total Activities
36
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Potent hFPRL1 (ALXR) agonists as potential anti-inflammatory agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 36 | 6.51 | 7.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL377226 | — | — | 1 | 7.64 |
| CHEMBL208884 | — | — | 1 | 7.52 |
| CHEMBL379762 | — | — | 1 | 7.52 |
| CHEMBL211220 | — | — | 1 | 7.37 |
| CHEMBL380389 | — | — | 1 | 7.36 |
| CHEMBL379761 | — | — | 1 | 7.36 |
| CHEMBL210303 | — | — | 1 | 7.10 |
| CHEMBL211957 | — | — | 1 | 7.09 |
| CHEMBL211595 | — | — | 1 | 7.08 |
| CHEMBL377969 | — | — | 1 | 7.05 |
| CHEMBL378064 | — | — | 1 | 7.00 |
| CHEMBL211885 | — | — | 1 | 7.00 |
| CHEMBL209995 | — | — | 1 | 6.85 |
| CHEMBL211555 | — | — | 1 | 6.82 |
| CHEMBL214216 | — | — | 1 | 6.77 |
| CHEMBL379853 | — | — | 1 | 6.60 |
| CHEMBL212113 | — | — | 1 | 6.51 |
| CHEMBL210298 | — | — | 1 | 6.31 |
| CHEMBL377130 | — | — | 1 | 6.27 |
| CHEMBL378679 | — | — | 1 | 6.11 |
| CHEMBL212109 | — | — | 1 | 6.01 |
| CHEMBL450023 | — | — | 1 | 5.90 |
| CHEMBL210475 | — | — | 1 | 5.83 |
| CHEMBL377642 | — | — | 1 | 5.56 |
| CHEMBL212116 | — | — | 1 | 5.43 |
| CHEMBL378707 | — | — | 1 | 5.31 |
| CHEMBL377163 | — | — | 1 | 5.29 |
| CHEMBL209102 | — | — | 1 | 5.23 |
| CHEMBL380160 | — | — | 1 | 4.91 |
| CHEMBL209521 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL377226 | — | EC50 | = | 23.0 | nM | 7.64 |
| CHEMBL208884 | — | EC50 | = | 30.0 | nM | 7.52 |
| CHEMBL379762 | — | EC50 | = | 30.0 | nM | 7.52 |
| CHEMBL211220 | — | EC50 | = | 43.0 | nM | 7.37 |
| CHEMBL380389 | — | EC50 | = | 44.0 | nM | 7.36 |
| CHEMBL379761 | — | EC50 | = | 44.0 | nM | 7.36 |
| CHEMBL210303 | — | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL211957 | — | EC50 | = | 81.0 | nM | 7.09 |
| CHEMBL211595 | — | EC50 | = | 83.0 | nM | 7.08 |
| CHEMBL377969 | — | EC50 | = | 90.0 | nM | 7.05 |
| CHEMBL378064 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL211885 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL209995 | — | EC50 | = | 140.0 | nM | 6.85 |
| CHEMBL211555 | — | EC50 | = | 150.0 | nM | 6.82 |
| CHEMBL214216 | — | EC50 | = | 170.0 | nM | 6.77 |
| CHEMBL379853 | — | EC50 | = | 250.0 | nM | 6.60 |
| CHEMBL212113 | — | EC50 | = | 310.0 | nM | 6.51 |
| CHEMBL210298 | — | EC50 | = | 490.0 | nM | 6.31 |
| CHEMBL377130 | — | EC50 | = | 540.0 | nM | 6.27 |
| CHEMBL378679 | — | EC50 | = | 770.0 | nM | 6.11 |
| CHEMBL212109 | — | EC50 | = | 980.0 | nM | 6.01 |
| CHEMBL450023 | — | EC50 | = | 1260.0 | nM | 5.90 |
| CHEMBL210475 | — | EC50 | = | 1470.0 | nM | 5.83 |
| CHEMBL377642 | — | EC50 | = | 2730.0 | nM | 5.56 |
| CHEMBL212116 | — | EC50 | = | 3700.0 | nM | 5.43 |
| CHEMBL378707 | — | EC50 | = | 4850.0 | nM | 5.31 |
| CHEMBL377163 | — | EC50 | = | 5130.0 | nM | 5.29 |
| CHEMBL209102 | — | EC50 | = | 5880.0 | nM | 5.23 |
| CHEMBL380160 | — | EC50 | = | 12300.0 | nM | 4.91 |
| CHEMBL209521 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL378062 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL210526 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL208979 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL386527 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL377169 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL208831 | — | EC50 | > | 10000.0 | nM | - |