Assay Detail
Functional
CHEMBL870425
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Activity at delta opioid receptor by MVD assay
2
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Synthesis and evaluation of 3-aminopropionyl substituted fentanyl analogues for opioid activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.46 | 7.46 |
| Inhibition | 1 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL214022 | — | — | 1 | 7.46 |
| CHEMBL216239 | CARBOXYFENTANYL | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL214022 | — | IC50 | = | 34.9 | nM | 7.46 |
| CHEMBL216239 | CARBOXYFENTANYL | Inhibition | = | 1.0 | % | - |