Assay Detail
Binding
CHEMBL872389
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity towards mouse hippocampal membranes cannabinoid receptor 1 using [3H]SR-141,716A
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Potent cannabinergic indole analogues as radioiodinatable brain imaging agents for the CB1 cannabinoid receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 8.30 | 8.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL364266 | — | — | 1 | 8.89 |
| CHEMBL188 | WIN-552122 | — | 1 | 7.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL364266 | — | Ki | = | 1.3 | nM | 8.89 |
| CHEMBL188 | WIN-552122 | Ki | = | 20.0 | nM | 7.70 |