Assay Detail
Binding
CHEMBL874088
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity towards rat liver V1a receptor was determined using [3H]arginine vasopressin as radioligand
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Development of a novel class of cyclic hexapeptide oxytocin antagonists based on a natural product.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 6.43 | 6.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL127686 | — | — | 1 | 6.43 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL127686 | — | Ki | = | 370.0 | nM | 6.43 |