Assay Detail
Binding
CHEMBL876970
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Ability to displace [3H]HU-243 binding to cannabinoid receptor in synaptosomal membrane
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Two new unsaturated fatty acid ethanolamides in brain that bind to the cannabinoid receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 7.34 | 7.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL321585 | — | — | 1 | 7.46 |
| CHEMBL15848 | ANANDAMIDE | — | 1 | 7.28 |
| CHEMBL105429 | — | — | 1 | 7.27 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL321585 | — | Ki | = | 34.4 | nM | 7.46 |
| CHEMBL15848 | ANANDAMIDE | Ki | = | 52.0 | nM | 7.28 |
| CHEMBL105429 | — | Ki | = | 53.4 | nM | 7.27 |