Assay Detail
Functional
CHEMBL878182
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Compound was evaluated for the competitive antagonism of NKA-stimulated PI (phosphatidylinositol) turnover in hamster urinary bladder tissue using [3H]inositol as radioligand
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Cricetulus griseus |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
A new class of high affinity ligands for the neurokinin A NK2 receptor: psi (CH2NR) reduced peptide bond analogues of neurokinin A4-10.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 6.70 | 6.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL341015 | — | — | 1 | 6.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL341015 | — | Kd | = | 199.53 | nM | 6.70 |