Assay Detail
Binding
CHEMBL879274
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of [3H]QNB binding to CHO cells bearing transfected muscarinic acetylcholine receptor M3
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cricetulus griseus |
| Cell Type | CHO |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Crystal, solution, and molecular modeling structural properties and muscarinic antagonist activity of azaprophen.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 9.33 | 9.33 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL287868 | AZAPROPHEN | — | 1 | 9.33 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL287868 | AZAPROPHEN | Ki | = | 0.472 | nM | 9.33 |