Assay Detail
Binding
CHEMBL882464
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory constant against human recombinant Beta-1,4-galactosyltransferase I
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Rational design, synthesis, and characterization of novel inhibitors for human beta1,4-galactosyltransferase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.31 | 5.31 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1743884 | UDP-GALACTOSE | — | 1 | 5.31 |
| CHEMBL2368692 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1743884 | UDP-GALACTOSE | Ki | = | 4910.0 | nM | 5.31 |
| CHEMBL2368692 | — | Ki | = | 149000.0 | nM | - |